AR-M 1000390 hydrochloride, Tocris Bioscience™

Description

Low-internalizing δ agonist

Non-peptidic, low-internalizing δ-selective opioid receptor agonist; derivative of SNC 80 (Cat. No. 0764). Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.

Specifications

Chemical Identifiers

• CAS: 209808-47-9
• Molecular Formula: C23H29ClN2O
• Molecular Weight (g/mol): 384.948
• InChI Key: OTXTZCLQEGSAMW-UHFFFAOYSA-N
• Synonym: ar-m 1000390 hydrochloride, arm390 hydrochloride, arm-390hcl, n,n-diethyl-4-phenyl-4-piperidinylidenemethyl-benzamide hydrochloride, n,n-diethyl-4-phenyl piperidin-4-ylidene methyl benzamide hydrochloride, arm1000390 hydrochloride, n,n-diethyl-4-phenyl-4-piperidinylidenemethyl benzamide hydrochloride
• PubChem CID: 76848958
• IUPAC Name: N,N-diethyl-4-[phenyl(piperidin-4-ylidene)methyl]benzamide;hydrochloride
• SMILES: CCN(CC)C(=O)C1=CC=C(C=C1)C(=C2CCNCC2)C3=CC=CC=C3.Cl

• Quantity: 10 mg
• Formula Weight: 384.94
• Percent Purity: >97%
• Chemical Name or Material: AR-M 1000390 hydrochloride