BRL 44408 maleate, Tocris Bioscience™

Description

Selective α2A antagonist

BRL 44408 maleate is a selective α2A-adrenoceptor antagonist (Ki = 1.7 nM and 144.5 nM at α2A and α2B-adrenergic receptors respectively). Increases hippocampal noradrenalin release following systemic administration.

Specifications

Chemical Identifiers

• CAS: 681806-46-2
• Molecular Formula: C17H21N3O4
• Molecular Weight (g/mol): 331.372
• InChI Key: DDIQGSUEJOOQQQ-BTJKTKAUSA-N
• Synonym: brl-44408 maleate, brl 44408 maleate salt, 2-2h-1-methyl-1,3-dihydroisoindole methyl-4,5-dihydroimidazole maleate salt, brl-44408 maleate salt, brl 44408 maleate salt hplc, 2-4,5-dihydro-1h-imidazol-2-ylmethyl-1-methyl-1,3-dihydroisoindole; maleic acid, 1h-isoindole, 2-4,5-dihydro-1h-imidazol-2-yl methyl-2,3-dihydro-1-methyl-, 2z-2-butenedioate 1:1
• PubChem CID: 10382026
• IUPAC Name: (Z)-but-2-enedioic acid;2-(4,5-dihydro-1H-imidazol-2-ylmethyl)-1-methyl-1,3-dihydroisoindole
• SMILES: CC1C2=CC=CC=C2CN1CC3=NCCN3.C(=CC(=O)O)C(=O)O

• Quantity: 10 mg
• Formula Weight: 331.37
• Percent Purity: >98%
• Chemical Name or Material: BRL 44408 maleate