Tocris Bioscience™ CGP 71683 hydrochloride

Highly selective and potent non-peptide NPY Y5 receptor antagonist

Brand:  Tocris Bioscience™ 2199/10

Product Code. 18757227

Description

CGP 71683 hydrochloride is an extremely selective, non-peptide NPY Y5 receptor antagonist. Displays > 1000-fold selectivity over Y1, Y2 and Y4 receptors; IC50 values are 1.4, 2765, 7187 and 5637 nM at cloned rat Y5, Y1, Y2 and Y4 receptors respectively. Potently inhibits NPY-induced food intake following i.p. administration in diabetic, free-feeding and fasted rats.

Specifications

• Purity: >99%
• Product Type: CGP 71683 hydrochloride
• Inhibitors: CGP 71683 hydrochloride

• Quantity: 10 mg
• Molecular Weight (g/mol): 512.07

For Research Use Only