missing translation for 'onlineSavingsMsg'
Learn More
  1. Home
  2. Products
  3. Chemicals
  4. Organic compounds
  5. Organonitrogen Compounds
  6. N-arylamides
  7. Gavestinel, Tocris Bioscience™

Gavestinel, Tocris Bioscience™

Product Code. 18065772
Click to view available options
Quantity:
10 mg
50 mg
This item is not returnable. View return policy
This item is not returnable. View return policy

Description

Potent and selective glycine site antagonist; orally available and active in vivo

Highly potent and selective non-competitive antagonist acting at the strychnine-insensitive glycine binding site of the NMDA receptor-channel complex (Kd = 0.8 nM). Displays > 1000-fold selectivity over NMDA, AMPA and kainate binding sites. Orally bioavailable and active in vivo.

Chemical Identifiers

CAS 153436-38-5
Molecular Formula C18H12Cl2N2NaO3
Molecular Weight (g/mol) 398.195
InChI Key OBPMZHMRJJJUBC-UHDJGPCESA-N
Synonym gavestinel
PubChem CID 67241466
IUPAC Name 3-[(E)-3-anilino-3-oxoprop-1-enyl]-4,6-dichloro-1H-indole-2-carboxylic acid;sodium
SMILES C1=CC=C(C=C1)NC(=O)C=CC2=C(NC3=CC(=CC(=C32)Cl)Cl)C(=O)O.[Na]

Specifications

Quantity 50 mg
Formula Weight 397.19
Percent Purity >98%
Chemical Name or Material Gavestinel
Product Content Correction

Your input is important to us. Please complete this form to provide feedback related to the content on this product.

Product Title

By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.

Thank You! Your feedback has been submitted. Fisher Scientific is always working to improve our content for you. We appreciate your feedback.