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GSK 269962, Tocris Bioscience™
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Quantity:
10 mg
50 mg
Description
Potent Rho kinase (ROCK) inhibitor (IC50 values are 1.6 and 4 nM for recombinant human ROCK1 and ROCK2 respectively). Displays greater than 30-fold selectivity for ROCK against a panel of serine/threonine kinases. Induces vasorelaxation in preconstricted rat aorta (IC50 = 35 nM); lowers blood pressure in a rat model of hypertension.
Specifications
Specifications
Quantity | 10 mg |
Formula Weight | 570.6 |
Percent Purity | >99% |
Chemical Name or Material | GSK 269962 |
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