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LEI 101 hydrochloride, Tocris Bioscience™

Catalog Number 30000735
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Quantity:
10 mg
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Description

Potent and selective CB2 partial agonist; orally biovailable

Potent and selective CB2 partial agonist (pEC50 = 8.0). Exhibits >100-fold selectivity for CB2 over CB1 and no significant interaction with hFAAH, MAGL, DAGL or NAPE-PLD. Displays antinociceptive activity in a rat neuropathic pain model and attenuates renal inflammation in a mouse kidney damage model. Orally bioavailable with low brain penetration.
CAS 2250025-91-1
Linear Formula C23H25FN4O4S.HCl
Quantity 10 mg
Synonym LEI 101 hydrochloride
Solubility Information Soluble to 100mM in DMSO
Formula Weight 508.99
Physical Form Solid
Chemical Name or Material 3-Cyclopropyl-1-[[4-[6-[(1,1-dioxido-4-thiomorpholinyl)methyl]-5-fluoro-2-pyridinyl]phenyl]methyl]-2
Grade >98%
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