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Tocris Bioscience™ MM 102

WDR5/MLL interaction inhibitor

Brand:  Tocris Bioscience™ 5307/10

Additional Details : Weight : 0.00970kg

Product Code. 18793968

  • £198.70 / 10mg
Estimated Shipment: 29-07-2024
to see stock.

Description

Description

MM 102 is a potent WDR5/MLL interaction inhibitor (IC50 = 2.4 nM). Inhibits MLL1 methyltransferase activity and MLL-1-induced HoxA9 and Meis-1 gene expression in leukemia cells expressing the MLL1-AF9 fusion gene. Also inhibits cell growth and induces apoptosis in leukemia cells harbouring MLL1 fusion proteins.
Specifications

Specifications

>98%
MM 102
MM 102
1883545-52-5
783.83
10 mg
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