Tocris Bioscience™ MRS 1220

Highly potent and selective hA3 antagonist

Brand:  Tocris Bioscience™ 1217/5

Product Code. 18757366

Description

A potent and highly selective antagonist at the human A3 adenosine receptor (Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. Displays an IC50 value > 1 μM for inhibition of binding to rat A3 receptors).

Specifications

• Quantity: 5 mg
• Assay: >98%
• Molecular Formula: C₂₁H₁₄ClN₅O₂
• Synonym: N-[9-Chloro-2-(2-furanyl)[1,2,4]-triazolo[1,5-c]quinazolin-5-yl]benzene acetamide
• Form: Solid

• Content And Storage: Store at room temperature
• CAS: 183721-15-5
• Formula Weight: 403.83
• Product Type: MRS 1220