NNC 26-9100, Tocris Bioscience™

Description

Selective sst4 agonist

NNC 26-9100 is a somatostatin sst4 receptor agonist that displays > 100-fold selectivity over sst2 receptors (Ki values are 6 and 621 nM for sst4 and sst2 receptors respectively). Potently inhibits forskolin -induced cAMP accumulation (EC50 = 26 nM).

Specifications

• CAS: 199522-35-5
• Molecular Formula: C22H25BrCl2N6S
• Quantity: 10 mg
• Synonym: 1-3-n-5-bromopyridin-2-yl-n-3,4-dichlorobenzyl amino propyl-3-3-1h-imidazol-4-yl propyl thiourea, 1-3-5-bromo-pyridin-2-yl-3,4-dichloro-benzyl-amino-propyl-3-3-1h-imidazol-4-yl-propyl-thiourea, 1-3-5-bromopyridin-2-yl 3,4-dichlorophenyl methyl amino propyl-3-3-1h-imidazol-4-yl propyl thiourea, thiourea,n-3-5-bromo-2-pyridinyl 3,4-dichlorophenyl methyl amino propyl-n'-3-1h-imidazol-5-yl propyl
• InChI Key: UREJDUPKGMFJRU-UHFFFAOYSA-N
• SMILES: C1=CC(=C(C=C1CN(CCCNC(=S)NCCCC2=CN=CN2)C3=NC=C(C=C3)Br)Cl)Cl
• IUPAC Name: 1-[3-[(5-bromopyridin-2-yl)-[(3,4-dichlorophenyl)methyl]amino]propyl]-3-[3-(1H-imidazol-5-yl)propyl]thiourea
• Molecular Weight (g/mol): 556.348
• PubChem CID: 9893924
• Formula Weight: 556.35
• Percent Purity: >99%
• Chemical Name or Material: NNC 26-9100