RJR 2403 oxalate, Tocris Bioscience™

Description

α4β2 selective nicotinic agonist

A neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki values are 26 and 36000 nM for α4β2 and α7 receptors respectively). Active in vivo.

Specifications

Chemical Identifiers

• CAS: 220662-95-3
• Molecular Formula: C12H16N2O4
• Molecular Weight (g/mol): 252.27
• InChI Key: WTIZFOAIQXMQHC-DPZBITMOSA-N
• Synonym: rjr-2403 oxalate, oxalic acid; rivanicline, e-n-methyl-4-3-pyridinyl-3-buten-1-amine oxalate, e-n-methyl-4-3-pyridinyl-3-bute n-1-amine oxalate, e-n-methyl-4-pyridin-3-yl but-3-en-1-amine oxalate, e-metanicotine oxalate;rivanicline oxalate;rjr 2403 oxalate, oxalic acid-3e-n-methyl-4-pyridin-3-yl but-3-en-1-amine 1/1
• PubChem CID: 23298272
• IUPAC Name: (E)-N-methyl-4-pyridin-3-ylbut-3-en-1-amine;oxalic acid
• SMILES: CNCCC=CC1=CN=CC=C1.C(=O)(C(=O)O)O

• Quantity: 50 mg
• Formula Weight: 252.27
• Percent Purity: >99%
• Chemical Name or Material: RJR 2403 oxalate