Tocris Bioscience™ SGC GAK 1

High affinity cyclin G associated kinase (GAK) inhibitor

Brand:  Tocris Bioscience™ 6564/25

Product Code. 18715348

Description

SGC GAK 1 is a high affinity cyclin G associated kinase (GAK) inhibitor (Kd = 1.9 nM). Exhibits >30-fold selectivity for GAK over a panel of other kinases. Inhibits GAK in live cell assays (IC50 = 110 nM).

Specifications

• Chemical Name or Material: 6-Bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine
• Quantity: 25 mg
• Purity: 99%

• CAS: 2226517-76-4
• Molecular Formula: C₁₈H₁₇BrN₂O₃