Tocris Bioscience™ Xanomeline oxalate

Functionally selective M1 agonist

Brand:  Tocris Bioscience™ 3569/10

Product Code. 18025322

Description

Xanomeline oxalate is a functionally selective muscarinic M1 receptor agonist (EC50 values are 0.3, 5, 42, 52 and 92.5 nM at M1, M3, M5, M4 and M2 receptors respectively). Displays a complex pharmacological profile: reversible and wash-resistant binding, resulting in full agonist activity at M1; delayed wash-resistant partial agonist activity at M2; and delayed wash-resistant full agonist activity at M4. Exhibits antipsychotic activity, and improves cognitive deficits and behavioral disturbances in Alzheimer's disease and schizophrenia.

Specifications

• Purity: >98%
• Product Type: Xanomeline oxalate
• Inhibitors: Xanomeline oxalate

• Quantity: 10 mg
• Molecular Weight (g/mol): 371.46

For Research Use Only