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Tocris Bioscience™ Perlapine
Potent muscarinc DREADD agonist
Brand: Tocris Bioscience™ 5549/10
This item is not returnable.
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Description
Perlapine is a potent muscarinic DREADD agonist (pEC50 values are 8.38, 8.08 and 7.27 for hM1Dq, hM3Dq and hM4Di in vitro, respectively). Exhibits >10,000-fold selectivity for hM3Dq over hM3 receptors.Specifications
6-(4-Methyl-1-piperazinyl)-11 H-dibenz[b,e]azepine | |
10 mg | |
C19H21N3 | |
99% |
1977-11-3 | |
DREADD Activators | |
291.39 |