Tocris Bioscience™ SET 2

Selective TRPV2 antagonist

Brand:  Tocris Bioscience™ 6990/10

Product Code. 18034142

Description

SET 2 is a TRPV2 (transient receptor potential vanilloid type 2) antagonist (IC50 = 0.46 μM). Selective for TRPV2 over TRPV1, TRPV3 and TRPV4 expressed in HEK293 cells. Inhibits lyosphosphatidic acid (LPA)-induced prostate cancer cell migration in vitro.

Specifications

• Chemical Name or Material: N-(2-Furanylmethyl)-3-[[4-(methylpropylamino)-6-(trifluoromethyl)-2-pyrimidinyl]thio]propanamide
• Quantity: 10 mg
• Molecular Formula: C₁₇H₂₁F₃N₄O₂S

• CAS: 2313525-20-9
• Target: TRPV Antagonists
• Purity: 0.98