Tocris Bioscience™ TASP 0390325

Potent and selective V1B receptor antagonist; orally bioavailable

Brand:  Tocris Bioscience™ 5729/50

Product Code. 18720118

Description

TASP 0390325 is a potent and selective V1B receptor antagonist (IC50 = 2.22 nM for rat pituitary receptor). Exhibits no significant affinity for 85 other receptors, ion channels and transporters at 10 μM, including V1A and V2. Increases ACTH levels in rats. Orally bioavailable. Antidepressant and anxiolytic.

Specifications

• Product Type: Antagonist
• CAS: 1642187-96-9
• Formula Weight: 554.44g/mol
• For Use With (Application): Vasopressin Receptor Antagonists

• Target Proteins: Vasopressin Receptor
• Molecular Formula: C₂₅H₂₉ClFN₅O₄.HCl
• Content And Storage: Store at -20°C
• Quantity: 50 mg

For Research Use Only