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Tocris Bioscience™ HC 067047
Potent and selective TRPV4 antagonist
£167.11 - £652.93
Specifications
Chemical Name or Material | 2-Methyl-1-[3-(4-morpholinyl)propyl]-5-phenyl-N-[3-(trifluoromethyl)phenyl]-1H-pyrrole-3-carboxamide |
---|---|
CAS | 883031-03-6 |
Target | TRPV Antagonists |
Molecular Formula | C26H28F3N3O2 |
Purity | 0.99 |
Product Code | Brand | Quantity | Price | Quantity & Availability | |||||
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Product Code | Brand | Quantity | Price | Quantity & Availability | |||||
18045232
|
Tocris Bioscience™
4100/50 |
50 mg |
£652.93
50mg |
Estimated Shipment: 20-08-2024 Log in to see stock. |
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18015432
|
Tocris Bioscience™
4100/10 |
10 mg |
£167.11
10mg |
Estimated Shipment: 20-08-2024 Log in to see stock. |
Please sign in to purchase this item. Need a web account? Register with us today! | ||||
Description
HC 067047 is a potent and selective TRPV4 antagonist. Reversibly inhibits currents through mouse, human and rat TRPV4 orthologs (IC50 values are 17, 48 and 133 nM respectively). Also inhibits the endogenous TRPV4-mediated response to 4α-PDH (IC50 = 22 nM). Selective for TRPV4 over TRPV1, TRPV2, TRPV3 and TRPM8 channels.Specifications
2-Methyl-1-[3-(4-morpholinyl)propyl]-5-phenyl-N-[3-(trifluoromethyl)phenyl]-1H-pyrrole-3-carboxamide | |
TRPV Antagonists | |
0.99 |
883031-03-6 | |
C26H28F3N3O2 |